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Pure Appl. Chem. Vol. 76, No. 5, pp. 907-1082 (2004)

Pure and Applied Chemistry

Vol. 76, Issue 5


Medicinal Chemistry

IUPAC Recommendations and Technical Reports

Lectures presented at the Polish-Austrian-German-Hungarian-Italian Joint Meeting on Medicinal Chemistry, Kraków, Poland, 15-18 October 2003

Preface, K. Kiec-Kononowicz and B. Malawska

Predicting drug metabolism: Concepts and challenges
B. Testa, A.-L. Balmat, and A. Long
p. 907 [Abstract] [full text - pdf 203KB]

Prion protein as a target for therapeutic interventions
P. P. Liberski
p. 915 [Abstract] [full text - pdf 176KB]

Structural basis for 2-amino-3-(3-hydroxy-5-methyl-4-isoxazolyl)propionic acid (AMPA) receptor activation
T. N. Johansen, J. R. Greenwood, S. B. Vogensen, and P. Krogsgaard-Larsen
p. 921 [Abstract] [full text - pdf 456KB]

Search for noncompetitive 2-amino-3-(3-hydroxy-5-methyl-4-isoxazolyl)propionic acid receptor (AMPAR) antagonists: Synthesis, pharmacological properties, and computational studies
A. Chimirri, G. De Sarro, S. Quartarone, M. L. Barreca, R. Caruso, L. De Luca, and R. Gitto
p. 931 [Abstract] [full text - pdf 382KB]

Neuropeptide mimetics for pain management
A. W. Lipkowski, A. Misicka, D. B. Carr, G. Ronsisvalle, D. Kosson, and I. Maszczynska Bonney
p. 941 [Abstract] [full text - pdf 281KB]

New endomorphin analogs with mu-agonist and delta-antagonist properties
G. Tóth, A. Keresztes, Cs. Tömböly, A. Péter, F. Fülöp, D. Tourwé, E. Navratilova, É. Varga, W. R. Roeske, H. I. Yamamura, M. Szucs, and A. Borsodi
p. 951 [Abstract] [full text - pdf 209KB]

Spacer conformation in biologically active molecules
J. Karolak-Wojciechowska and A. Fruzinski
p. 959 [Abstract] [full text - pdf 244KB]

Discovery of new anti-inflammatory agents
F. Fülöp, L. Lázár, Z. Szakonyi, M. Pihlavisto, S. Alaranta, P. J. Vainio, A. Juhakoski, A. Marjamäki, and D. J. Smith
p. 965 [Abstract] [full text - pdf 239KB]

NO donors: Focus on furoxan derivatives
A. Gasco, R. Fruttero, G. Sorba, A. Di Stilo, and R. Calvino
p. 973 [Abstract] [full text - pdf 246KB]

Passive and catalytic antibodies and drug delivery
G. M. Blackburn, J. H. Rickard, S. Cesaro-Tadic, D. Lagos, A. Mekhalfia, L. Partridge, and A. Plückthun
p. 983 [Abstract] [full text - pdf 255KB]

Virtual combinatorial chemistry and in silico screening: Efficient tools for lead structure discovery?
T. Langer and G. Wolber
p. 991 [Abstract] [full text - pdf 148KB]

Development of modulators of multidrug resistance: A pharmacoinformatic approach
G. F. Ecker and P. Chiba
p. 997 [Abstract] [full text - pdf 269KB]

Hindered nucleoside analogs as antiflaviviridae agents
S. Manfredini, A. Angusti, A. C. Veronese, E. Durini, S. Vertuani, F. Nalin, N. Solaroli, S. Pricl, M. Ferrone, M. Mura, M. A. Piano, B. Poddesu, A. Cadeddu, P. La Colla, and R. Loddo
p. 1007 [Abstract] [full text - pdf 297KB]

Solid- and solution-phase synthesis of bioactive dihydropyrimidines
D. Dallinger, A. Stadler, and C. O. Kappe
p. 1017 [Abstract] [full text - pdf 245KB]

Synthesis of naturally occurring o-heterocyclic compounds of biological activity
S. Antus, K. Gulácsi, L. Juhász, L. Kiss, and T. Kurtán
p. 1025 [Abstract] [full text - pdf 299KB]


IUPAC Recommendations and Technical Reports

Glossary of terms used in toxciokinetics (IUPAC Recommendations 2003)
M. Nordberg, J. Duffus, and D. M. Templeton
p. 1033 [Abstract] [full text - pdf 319KB]


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